کد مقاله کد نشریه سال انتشار مقاله انگلیسی نسخه تمام متن
7806958 1501646 2018 14 صفحه PDF دانلود رایگان
عنوان انگلیسی مقاله ISI
Novel trifluoromethylpyrazole acyl urea derivatives: Synthesis, crystal structure, fungicidal activity and docking study
ترجمه فارسی عنوان
مشتقات تری فلوئور متیل پیازولول آکریل اوره: سنتز، ساختار بلوری، فعالیت قارچ کش و مطالعه اتصال
کلمات کلیدی
تری فلوئور متیل پیازول، اوره، فعالیت قارچ کش، دوختن سنتز،
موضوعات مرتبط
مهندسی و علوم پایه شیمی شیمی آلی
چکیده انگلیسی
Thirteen novel trifluoromethylpyrazole acyl urea derivatives were designed and synthesized. In vivo fungicidal activities of these compounds were tested against Fusarium oxysporum, Corynespora mazei, Botrytis cinerea and Pseudomonas syringae respectively, particularly compounds exhibited significant control effective at 100 mg/L. More importantly, some compounds showed the good control effective at 10 mg/L. Furthermore, docking was established to study the structure-activity relationship of the title compounds. It is possible that trifluoromethylpyrazole acyl urea derivatives, which possess good control effective against Fusarium oxysporum, Corynespora mazei and Botrytis cinerea, may become novel lead compounds for the development of fungicides with further structure modification.
ناشر
Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Journal of Molecular Structure - Volume 1171, 5 November 2018, Pages 631-638
نویسندگان
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