Development of novel amide-derivatized 2,4-bispyridyl thiophenes as highly potent and selective Dyrk1A inhibitors. Part II: Identification of the cyclopropylamide moiety as a key modification

Physical Sciences and Engineering Chemistry Organic Chemistry

Sarah S. Darwish, Mohammad Abdel-Halim, Ahmed K. ElHady, Mohamed Salah, Ashraf H. Abadi, Walter Becker, Matthias Engel,