Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5158727 | European Journal of Medicinal Chemistry | 2017 | 84 Pages |
Abstract
Aiming to develop potent agonist with improved efficacy and safety, we have identified series of FFA1 agonists bearing sulfone-carboxylic acid moiety, exemplified by the potent and orally bioavailable agonist 20.322
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Zheng Li, Chunxia Liu, Xue Xu, Qianqian Qiu, Xin Su, Yuxuan Dai, Jianyong Yang, Huilan Li, Wei Shi, Chen Liao, Miaobo Pan, Wenlong Huang, Hai Qian,