Article ID Journal Published Year Pages File Type
5213188 Tetrahedron 2016 5 Pages PDF
Abstract

The palladium-catalyzed three-component cycloaminocarbonylation of 2-formylaryl tosylates with hydrazines and carbon monoxide has been established, which provides an efficient method for synthesis of substituted phthalazinones. In addition, by applying this protocol as the key step, Hydralazine can easily be synthesized in 65% yield.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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