| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5213334 | Tetrahedron | 2016 | 5 Pages |
Abstract
A novel dehydrodimerization of malonates with indoles has been developed, providing simple and rapid access to 3-indolyl tetramethyl 1,1,2,2-ethanetetracarboxylates. Pd(OAc)2-catalyzed ‘one pot’ C(sp2)–C(sp3) and C(sp3)–C(sp3) cross-dehydrogenative-couplings of malonates with a variety of 2-aryl indoles were involved. The titled compounds were obtained in high yields with good functional group tolerance.
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Related Topics
Physical Sciences and Engineering
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