Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5213503 | Tetrahedron | 2016 | 8 Pages |
Abstract
A convenient and regioselective cross-coupling of heteroaryl boronic acids with allylic alcohols under catalyst-free reaction conditions is described. The developed procedure is simple, works under external oxidant- and metal-free conditions, and proves to be very general with an unprecedented ortho-selectivity. This approach represents one of the very few examples of ortho-functionalization of boronic acids.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Xue-Dong Li, Li-Jun Xie, De-Long Kong, Li Liu, Liang Cheng,