| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5213740 | Tetrahedron | 2016 | 6 Pages |
Abstract
The conventional etherification uses toxic or hardly degradable alkylating agents. An eco-friendly tandem etherification/aromatization is presented to prepare estrone 3-secondary ethers from easily available dienone 1. Three marketed 3-etherified estrogen drugs were synthesized with the method from commercial available starting material.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Dong-Qing Zheng, Yu Jing, Bing-Ying Zheng, Yun-Fei Ye, Sheng Xu, Wei-Sheng Tian, Hai-Yan Ma, Kai Ding,