| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5215072 | Tetrahedron | 2015 | 9 Pages |
Abstract
A series of substituted indoloquinolinones were readily synthesized, via two steps, from indole-2-carboxylic acid and its derivatives: a 3-arylation of indole-2-carboxamides and a subsequent PIDA-mediated oxidative C-N bond formation. The underpinning strategy involves a Cu(I)-promoted C(sp2)-C(sp2) coupling and a PIDA-mediated oxidative C(sp2)-N coupling.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Yulin Li, Daisy Zhang-Negrerie, Yunfei Du, Kang Zhao,