Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5215446 | Tetrahedron | 2014 | 9 Pages |
Abstract
A total synthesis of Daphnodorin A, a member of the Daphnodorins, was accomplished. Key features of the synthetic strategy include construction of 2-substituted-3-functionalized benzofuran via intramolecular Heck reaction and a mild Barton-McCombie deoxygenation process mediated by triethylborane. The total synthesis provided Daphnodorin A in 19.7% or 5.6% overall yield over 7 or 15 steps.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Hu Yuan, Kaijian Bi, Wanlin Chang, Rongcai Yue, Bo Li, Ji Ye, Qingyan Sun, Huizi Jin, Lei Shan, Weidong Zhang,