Article ID Journal Published Year Pages File Type
5215807 Tetrahedron 2014 4 Pages PDF
Abstract

A copper-catalyzed thiolation annulation of o-halostyrenes with sodium hydrosulfide has been developed. In the presence of Cu(OTf)2 and 1,4-benzoquinone, a variety of 2-substituted benzothiophenes were prepared in moderate to good yields by tandem C-S bond forming reaction and hydrothiolation of olefins.

Graphical abstractDownload full-size image

Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
Authors
, , , , ,