Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5215961 | Tetrahedron | 2014 | 6 Pages |
Abstract
A general and efficient strategy for fused tricyclic indoles from substituted 2-halogenanilines via the palladium-catalyzed intramolecular Larock indolization process has been developed. Using this strategy, a number of 3,4- and 3,5-fused indoles with a variety of ring sizes can been prepared. The utility of this method is demonstrated through the synthesis of the known tetrahydropyrrolo[4,3,2-de]quinoline 10 and the first total synthesis of fargesine.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Yan Gao, Dong Shan, Yanxing Jia,