| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5216232 | Tetrahedron | 2014 | 8 Pages |
Abstract
An efficient protocol was developed for regio-selective Pd-catalyzed direct ortho-fluorination of 2-arylbenzo[d]thiazoles using N-fluorobenzenesulfonimide (NFSI) as the F+ source, and l-proline as the crucial promoter. The present method offered a practical route to synthesize valuable fluorinated products, which are of potential importance in the pharmaceutical and agrochemical industries.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Qiuping Ding, Changqing Ye, Shouzhi Pu, Banpeng Cao,