Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5216570 | Tetrahedron | 2014 | 5 Pages |
Abstract
A novel Pd(II)-catalyzed dehydrogenative cross-coupling reaction of thiazolo[5,4-d]pyrimidine with unactivated (hetero)arenes via C-H bond activation was achieved. This protocol provides a straightforward and operationally simple method for the synthesis of 2-arylsubstituted thiazolo[5,4-d]pyrimidines of interest in pharmaceutical sciences.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Sheng-Wei Yang, Ye-Xiang Su, Li-Ping Sun,