Article ID Journal Published Year Pages File Type
5216570 Tetrahedron 2014 5 Pages PDF
Abstract

A novel Pd(II)-catalyzed dehydrogenative cross-coupling reaction of thiazolo[5,4-d]pyrimidine with unactivated (hetero)arenes via C-H bond activation was achieved. This protocol provides a straightforward and operationally simple method for the synthesis of 2-arylsubstituted thiazolo[5,4-d]pyrimidines of interest in pharmaceutical sciences.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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