Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5216664 | Tetrahedron | 2014 | 9 Pages |
Abstract
The direct imine acylation (DIA) and subsequent cyclisation of a range of imines with ortho-substituted benzoic acid derivatives is described. Variation in the coupling reagents, imine and benzoic acid were all examined. The DIA procedure was also applied in the total synthesis of (±)-cavidine.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Christiana Kitsiou, William P. Unsworth, Graeme Coulthard, Richard J.K. Taylor,