| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5217374 | Tetrahedron | 2013 | 6 Pages |
Abstract
The synthesis of fused thiophene-cyclopentanes by PdII-catalyzed dehydrogenative C(sp2)-H/C(sp3)-H coupling is described. This reaction shows interesting chemo- and diastereoselectivity, however a direct comparison showed that it is yet much less efficient than the two-step sequence composed of electrophilic halogenation and Pd0-catalyzed C(sp3)-H arylation.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Cathleen Pierre, Olivier Baudoin,