| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5217533 | Tetrahedron | 2013 | 7 Pages |
Abstract
A novel three-step approach leading to [1,2,3]-triazolo[1,5-a][1,4]benzodiazepines in moderate to good yields has been developed. The key step is an unprecedented one-pot Cu-catalyzed azidation-cyclization reaction of ortho-bromobenzylpropargylamines.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
![Synthesis of [1,2,3]-triazolo[1,5-a][1,4]benzodiazepines via an unprecedented one-pot Cu-catalyzed azidation-cyclization reaction](/preview/png/5217533.png "First Page Preview: Synthesis of [1,2,3]-triazolo[1,5-a][1,4]benzodiazepines via an unprecedented one-pot Cu-catalyzed azidation-cyclization reaction")
Authors
Geert Hooyberghs, Hendrik De Coster, Dipak D. Vachhani, Denis S. Ermolat'ev, Erik V. Van der Eycken,