Article ID Journal Published Year Pages File Type
5218048 Tetrahedron 2013 4 Pages PDF
Abstract

Tetraethylenepentamine and triethylenetetramine are found to be efficient organic bases for the N-arylation of pyrazole and imidazole with aryl and heteroaryl-iodides and -bromides catalyzed by CuI in water at moderate temperature. The cross-couplings proceed smoothly with good to excellent yields and a variety of functional groups are tolerated under this condition.

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Physical Sciences and Engineering Chemistry Organic Chemistry
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