Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5218048 | Tetrahedron | 2013 | 4 Pages |
Abstract
Tetraethylenepentamine and triethylenetetramine are found to be efficient organic bases for the N-arylation of pyrazole and imidazole with aryl and heteroaryl-iodides and -bromides catalyzed by CuI in water at moderate temperature. The cross-couplings proceed smoothly with good to excellent yields and a variety of functional groups are tolerated under this condition.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Qichao Yang, Yufang Wang, Li Yang, Mingjie Zhang,