Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5218051 | Tetrahedron | 2013 | 11 Pages |
Abstract
Starting from phthalimidoalkanoylamines 1 (amino-protected derivatives of glycine, β-alanine, γ-amino butyric, δ-amino valeric, and ε-amino caproic acids), a facile synthetic method has been developed to obtain diethyl 5-alkyl(dialkyl)amino-2-aminoalkyl-1,3-oxazol-4-ylphosphonates 7, which have been further used in the preparation of phosphorylated peptidomimetics 10 and 12.
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Chemistry
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Authors
Kostyantyn M. Kondratyuk, Olena I. Lukashuk, Aleksandr V. Golovchenko, Igor V. Komarov, Volodymyr S. Brovarets, Valery P. Kukhar,