Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5218315 | Tetrahedron | 2013 | 7 Pages |
Abstract
An In(OTf)3-catalyzed N-benzylation of amines utilizing benzyl alcohols through direct C-O bond activation has been reported. The reaction was performed in water without any base, additive, ligand or inert gas protection to afford the chem-selective mono- or bis-alkylated aromatic amines in good to excellent yields.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Jin-Ming Yang, Ran Jiang, Lin Wu, Xiao-Ping Xu, Shun-Yi Wang, Shun-Jun Ji,