Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5218351 | Tetrahedron | 2012 | 5 Pages |
Abstract
Highly important trans-3,4-dihydro-2H-1,4-benzoxazine moieties were easily synthesized by domino aziridine ring opening with o-bromophenols and o-chlorophenols followed by the palladium catalyzed coupling-cyclization (intramolecular C(aryl)-N(amide) bond formation) with good to excellent yields.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
R. Koteshwar Rao, I. Karthikeyan, Govindasamy Sekar,