| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5218357 | Tetrahedron | 2012 | 8 Pages |
Abstract
A two-step sequence is reported giving access to diverse 5H-pyrido[2â²,1â²:2,3]imidazo[4,5-b]indoles and analogues via a Bienaymé multicomponent reaction followed by N-arylation. The desired polycylic scaffolds were obtained in high yield using copper iodide in association with TMEDA in aqueous or dioxane media.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
![Straightforward Bienaymé and copper catalyzed N-arylation sequence to access diverse 5H-pyrido[2â²,1â²:2,3]imidazo[4,5-b]indoles and analogues](/preview/png/5218357.png "First Page Preview: Straightforward Bienaymé and copper catalyzed N-arylation sequence to access diverse 5H-pyrido[2â²,1â²:2,3]imidazo[4,5-b]indoles and analogues")
Authors
Ahmed El Akkaoui, Marie-Aude Hiebel, Abderrahim Mouaddib, Sabine Berteina-Raboin, Gérald Guillaumet,