| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5218388 | Tetrahedron | 2013 | 7 Pages |
Abstract
A facile and efficient way for the synthesis of the acylated 2-arylbenzoxazoles and 2-arylbenzothiazoles by heterocycle-directed ortho-acylation was developed. This reaction was performed in chlorobenzene, using arylmethyl alcohols and tert-butyl hydroperoxide (TBHP) as the easily accessible acyl source and the oxidant, respectively, affording the desired products in moderate to good yields.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Qian Zhang, Fan Yang, Yangjie Wu,