| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5218617 | Tetrahedron | 2013 | 7 Pages |
Abstract
A gold-catalyzed regioselective heteroannulation strategy has been developed for the concise and efficient synthesis of imidazo[1,2-a]pyrazinones. The protocol allows the introduction of diversity via the application of substituted propargyl amines or via Suzuki-coupling of the generated imidazo[1,2-a]pyrazinones with various (het)aryl boronic acids.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
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Authors
Dipak D. Vachhani, Sachin G. Modha, Abhishek Sharma, Erik V. Van der Eycken,