Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5218706 | Tetrahedron | 2012 | 9 Pages |
Abstract
Practical and straightforward method for regioselective C-S bond formation accomplished by copper-catalyzed regioselective C-F substitution of electron-deficient perfluoroarenes with aryl thioacetates or benzyl thioacetate has been developed. Because of its high reaction efficiency, good chemoselectivity and regioselectivity, and excellent functional-group compatibility, this protocol provides a useful and operationally simple access to polyfluoroaryl thioethers used for drugs and material chemistry.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Qizhong Zhou, Bin Zhang, Tieqi Du, Haining Gu, Huajiang Jiang, Rener Chen,