| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5219155 | Tetrahedron | 2013 | 6 Pages |
Abstract
The synthesis of 7-aminoacetylindoles was achieved via the hydrogenation of 7-acylcyanides, which were produced through the oxidation of indole-7-cyanohydrin silylether intermediates. 7-Oxotryptamines were subsequently converted into 5-(7â²-indolyl)oxazoles by reaction with acetic anhydride followed by phosphoryl chloride, and to 2,5-di-(7â²-indolyl)oxazoles by reaction with 7-trichloroacetylindoles followed by phosphoryl chloride.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Hakan Kandemir, Kasey Wood, Naresh Kumar, David StC. Black,