Article ID Journal Published Year Pages File Type
5219197 Tetrahedron 2012 7 Pages PDF
Abstract

d-Homotryptophan and its sulfur analogue have been synthesized by Sonogashira coupling between 3-iodoheteroarenes and ethynyloxazolidine followed by reduction of triple bond and oxidation of alcohol to acid. l-Homotryptophan and its oxygen analogue have been synthesized from silylated internal alkyne using Larock's heteroannulation as the key reaction. The alkynyloxazolidines were synthesized from l-serine and l-glutamic acid, respectively.

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Physical Sciences and Engineering Chemistry Organic Chemistry
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