| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5219343 | Tetrahedron | 2011 | 10 Pages |
Abstract
Substituted imidazoles and purine bioisosteres have been widely studied in the literature. We endeavored to combine these heterocyclic core structures into precursors, especially 7-azaindoles, of previously unknown pharmacologically relevant lead structures. A highly flexible synthetic procedure was developed, derived from investigations of the influence of the substrates, solvents, ligand systems, and side reactions.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Roland Selig, Dieter Schollmeyer, Wolfgang Albrecht, Stefan Laufer,