Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5219432 | Tetrahedron | 2012 | 7 Pages |
Abstract
Regioselective copper(I)-catalyzed C-H hydroxylation/C-S coupling of aryl thiols with vinyl halides was developed. Starting from substituted aryl thiols and vinyl halides, various 2-(styrylthio)phenol derivatives were efficiently prepared. The application of the synthetic methodology to generate the bioactive organic intermediate was also exemplified.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Run-Sheng Xu, Lei Yue, Yuan-Jiang Pan,