Article ID Journal Published Year Pages File Type
5219432 Tetrahedron 2012 7 Pages PDF
Abstract

Regioselective copper(I)-catalyzed C-H hydroxylation/C-S coupling of aryl thiols with vinyl halides was developed. Starting from substituted aryl thiols and vinyl halides, various 2-(styrylthio)phenol derivatives were efficiently prepared. The application of the synthetic methodology to generate the bioactive organic intermediate was also exemplified.

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Physical Sciences and Engineering Chemistry Organic Chemistry
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