Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5220084 | Tetrahedron | 2012 | 8 Pages |
Abstract
An intramolecular palladium(0)-mediated ortho-arylation of phenols applied to the synthesis of various substituted aporphines is reported. Most significantly, the efficiency of the transformation was enhanced by the use of monoligated Pd(0) complexes. This methodology was extended to para-arylation of phenols and employed in the synthesis of the aporphine alkaloid (â)-lirinine.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Malik Hellal, Shambhavi Singh, Gregory D. Cuny,