| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5221171 | Tetrahedron | 2012 | 5 Pages |
Abstract
(â)-Benzolactam-V8, an artificially-designed cyclic dipeptide with strong tumor-promoter activity, was synthesized from benzyl (S)-N-(2-formylphenyl)-N-methylvalinate by application of guanidinium ylide-participated asymmetric aziridination followed by the reductive ring-opening reaction of 3-arylaziridine-2-carboxylate formed.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Itsara Khantikaew, Masato Takahashi, Takuya Kumamoto, Noriyuki Suzuki, Tsutomu Ishikawa,