| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5221275 | Tetrahedron | 2010 | 7 Pages |
Abstract
A novel series of 4-aminobenzofused sultams was prepared using an efficient synthetic procedure based on superacid mediated reactions followed either by copper-catalyzed coupling or SNAr reactions. The synthetic potential of the method toward the divergent synthesis of novel potent bioactive (fluorinated) aminobenzofused sultams and fluorinated 4-aminobenzene sulfonamides was shown, making it a new valuable process to synthesize a large diversity of compounds in bioactive 4-aminobenzene sulfonamide family.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Fei Liu, Neil Y. Musadji, Frédéric Lecornué, Marie-Paule Jouannetaud, Sébastien Thibaudeau,