| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5221506 | Tetrahedron | 2012 | 5 Pages |
Abstract
A highly efficient palladium-catalyzed direct desulfitative arylation of azoles at C2-position has been developed using sodium arylsulfinates as aryl sources. Azoles including benzoxazoles, benzothiazoles, oxazoles, thiazoles, and 1,3,4-oxadiazoles reacted with sodium arylsulfinates smoothly to generate the corresponding products in good to excellent yields, and various substitution patterns were tolerated toward the reaction.
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Physical Sciences and Engineering
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