| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5221609 | Tetrahedron | 2011 | 6 Pages |
Abstract
A facile and environment-benign oxidation by dioxygen as the sole oxidant was applied for the conversion of 2-oxazolines to oxazoles. The substituent effect on 2-oxazoline ring was investigated. The use of this methodology for the synthesis of a key intermediate of a CDC25 phosphatase inhibitor (SC-ααδ9) as an anticancer agent was also described.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Yue Huang, Lijun Ni, Haifeng Gan, Yu He, Jinyi Xu, Xiaoming Wu, Hequan Yao,