| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5222565 | Tetrahedron | 2009 | 6 Pages |
Abstract
A series of non-peptidic HIV protease inhibitors were synthesized starting from the same optically active precursor, (S)-glycidol. The substrate was easily converted into different indolic sulfonamides or amines by regioselective reactions. The preliminary inhibitory activity was evaluated.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Lucia Chiummiento, Maria Funicello, Paolo Lupattelli, Francesco Tramutola, Pietro Campaner,