| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5222714 | Tetrahedron | 2011 | 7 Pages |
Abstract
Potentially bioactive 3-(anilinoarylmethylene)-2-oxindoles as Hesperadin analogoues have been synthesized via a two-step procedure: (a) an Ugi-4MCR and (b) reaction of the Ugi adduct with aniline in the presence of a palladium catalyst via domino Heck/Buchwald reaction. In all cases, a single isomer with the Z-configuration was obtained in good to high yields.
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