| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5222766 | Tetrahedron | 2010 | 8 Pages |
Abstract
A convenient synthesis of 1,2,3-triazole-fused isoindolines and dihydroisoquinolines in good to excellent yield is reported, starting from easily available terminal alkynes and (2-haloaryl)alkylazides. The method is based upon a cycloaddition reaction, via click chemistry, followed by a transition metal-catalyzed functionalization of a C-H bond.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Vito Fiandanese, Giuseppe Marchese, Angela Punzi, Francesco Iannone, Giacomo G. Rafaschieri,