Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5222866 | Tetrahedron | 2011 | 6 Pages |
Abstract
N-Alkoxymethylation of heterocyclic compounds with diethyl phosphite via cleavage of P–O bond was investigated and a series of N3-ethoxymethylated heterocyclic compounds were synthesized. A mechanism in which diethyl phosphite acts as an efficient surrogate of ethanol was proposed and supported by several evidences.
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