Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5223022 | Tetrahedron | 2011 | 6 Pages |
Abstract
A Brønsted acid catalyzed Diels–Alder reaction of 2-vinylindoles and 3-nitrocoumarins has been described. The methodology allows a rapid and expedient synthesis of a variety of coumarin-fused polycyclic indoles in good yields (up to 82%) with high diastereoselectivities (up to >19:1).
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