Article ID Journal Published Year Pages File Type
5223022 Tetrahedron 2011 6 Pages PDF
Abstract

A Brønsted acid catalyzed Diels–Alder reaction of 2-vinylindoles and 3-nitrocoumarins has been described. The methodology allows a rapid and expedient synthesis of a variety of coumarin-fused polycyclic indoles in good yields (up to 82%) with high diastereoselectivities (up to >19:1).

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry