Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5223226 | Tetrahedron | 2010 | 5 Pages |
Abstract
Copper-catalyzed amination of N-heterocycle derived aryl iodides followed by intramolecular condensative cyclization afforded N-substituted pyrrolo[2,1-c][1,4]-benzodiazepine-5,11-diones with good yields. By varying primary amines and substituents at aromatic ring of aryl iodides, a wide range of these heterocycles were assembled.
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Related Topics
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Chemistry
Organic Chemistry
Authors
Xu Lu, Liu Shi, Hui Zhang, Yongwen Jiang, Dawei Ma,