| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5223350 | Tetrahedron | 2009 | 6 Pages |
Abstract
In this paper, we describe the synthesis of conformationally constrained dipeptide mimetic derivatives. Microwave flash heating was used in several synthetic steps providing the opportunity to perform the reactions in dramatically shortened time as well as to increase the obtained yields. The efficiency of the methodology makes it useful in order to prepare other dipeptides containing the 4-amino-tetrahydro-2-benzazepin-3-one motif.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Beatrice Severino, Ferdinando Fiorino, Antonella Esposito, Francesco Frecentese, Francesca De Angelis, Elisa Perissutti, Giuseppe Caliendo, Vincenzo Santagada,