Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5223520 | Tetrahedron | 2010 | 6 Pages |
Abstract
Anodic fluorination of various N-acetyl-3-substituted indole derivatives was successfully carried out in Et4NF-4HF/MeCN to provide the corresponding trans-2,3-difluoro-2,3-dihydroindoles exclusively or selectively. Treatment of difluorinated products with a base provided monofluoroindole derivatives or monofluoroindoline derivative depending on the substituents at the 3-position.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Bin Yin, Laihao Wang, Shinsuke Inagi, Toshio Fuchigami,