Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5223853 | Tetrahedron | 2010 | 7 Pages |
Abstract
A series of trihalogenated alkenylbenzenes undergo consecutive palladium catalyzed inter- and intramolecular amination reactions to deliver a series of 1-functionalized mono-chloroindoles. 4-, 5-, 6- and 7-Chloroindoles can all be prepared; carbamates, anilines and amines can be employed as the N-nucleophile.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Luke C. Henderson, Matthew J. Lindon, Michael C. Willis,