| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5224082 | Tetrahedron | 2008 | 5 Pages |
Abstract
4-Allyl-phosphaisoquinolin-1-ones were synthesized by palladium-catalyzed coupling-cyclization of o-ethynylphenylphosphonamide monoethyl esters with allyl halides with high regioselectivity and good yields. The synthesized 4-allyl-phosphaisoquinolin-1-ones show bioactivity as inhibitor of MCH-1R.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Wei Tang, Yi Ding, Yi-Xiang Ding,