Article ID Journal Published Year Pages File Type
5224427 Tetrahedron 2009 4 Pages PDF
Abstract

The reaction of 2-(chloromethyl)phenyl isocyanides, readily available by dehydration of the respective N-[2-(chloromethyl)phenyl]formamides, with organolithiums produced 2-substituted indoles in satisfactory yields through addition of organolithiums to the isocyano carbon followed by intramolecular substitution reaction of the resulting imidoyl anion intermediates.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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