Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5224739 | Tetrahedron | 2008 | 9 Pages |
Abstract
Condensation of diphenylacetaldehydes and 1,1-diphenylacetones with malonodinitrile and cyclization of obtained aryl-ylidenemalonodinitriles in concentrated sulfuric acid leads to 1-amino-4-arylnaphthalene-2-carbonitriles. The benzannulation reaction is accompanied by a quasi-aromatic rearrangement. Preliminary tests of some synthesized aminonitriles have revealed their considerable biological activity against phytopathogenic fungi.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
BartÅomiej Kozik, JarosÅaw Wilamowski, Maciej Góra, Janusz J. SepioÅ,