Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5224838 | Tetrahedron | 2009 | 5 Pages |
Abstract
An efficient formal synthesis of S-(+) dapoxetine starting from 3-hydroxy azetidin-2-one is described. The intermediate (S)-3-(dimethyl amino)-3-phenylpropan-1-ol was synthesized in enantiopure form starting with 3-hydroxy azetidin-2-one in seven steps.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Pinak M. Chincholkar, Ajaykumar S. Kale, Vikas K. Gumaste, Abdul Rakeeb A.S. Deshmukh,