Article ID Journal Published Year Pages File Type
5224838 Tetrahedron 2009 5 Pages PDF
Abstract

An efficient formal synthesis of S-(+) dapoxetine starting from 3-hydroxy azetidin-2-one is described. The intermediate (S)-3-(dimethyl amino)-3-phenylpropan-1-ol was synthesized in enantiopure form starting with 3-hydroxy azetidin-2-one in seven steps.

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Physical Sciences and Engineering Chemistry Organic Chemistry
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