| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5224862 | Tetrahedron | 2008 | 8 Pages |
Abstract
Starting from a library of 2-l-α-amino acyl (E)-acrylonitriles, different short 2-cyano and 2-amido aziridinyl peptides, potential protease inhibitors, were obtained under parallel solution-phase conditions. The transformations include careful selection of conditions for aziridine deprotection and cyano group partial hydrolysis.
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Authors
Stefania Fioravanti, Davide Massari, Alberto Morreale, Lucio Pellacani, Paolo A. Tardella,