| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5225586 | Tetrahedron | 2009 | 6 Pages |
Abstract
An efficient and convergent one-step synthesis of substituted dihydroquinolin-2-ones from α,β-unsaturated esters and aminoaryl pinacolboronates under rhodium catalysis is reported. The reaction is easily applicable in parallel synthesis format and provides convenient access to this pharmaceutically-relevant motif.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Joachim Horn, Ho Yin Li, Stephen P. Marsden, Adam Nelson, Rachel J. Shearer, Amanda J. Campbell, David House, Gordon G. Weingarten,