Article ID Journal Published Year Pages File Type
5225710 Tetrahedron 2009 6 Pages PDF
Abstract

A general, efficient, and inexpensive method for the N-arylation of indoles using a catalytic system derived from CuI and benzotriazole is reported. Selective mono N-arylation of indoles with ortho-dihaloarenes has also been successfully achieved in good yields using this protocol.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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