Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5225710 | Tetrahedron | 2009 | 6 Pages |
Abstract
A general, efficient, and inexpensive method for the N-arylation of indoles using a catalytic system derived from CuI and benzotriazole is reported. Selective mono N-arylation of indoles with ortho-dihaloarenes has also been successfully achieved in good yields using this protocol.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Akhilesh Kumar Verma, Jaspal Singh, Richard C. Larock,