Article ID Journal Published Year Pages File Type
5226203 Tetrahedron 2009 6 Pages PDF
Abstract

The regioselective synthesis of halogenated aminopyrimidinyl-pyrroles as useful scaffolds for the preparation of diversified selective kinase inhibitors is described. The chemistry is simple and mostly based on the use of N-halosuccinimides under mild reaction conditions but the regioselectivity observed is partially unexpected.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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