Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5226203 | Tetrahedron | 2009 | 6 Pages |
Abstract
The regioselective synthesis of halogenated aminopyrimidinyl-pyrroles as useful scaffolds for the preparation of diversified selective kinase inhibitors is described. The chemistry is simple and mostly based on the use of N-halosuccinimides under mild reaction conditions but the regioselectivity observed is partially unexpected.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Ermes Vanotti, Marina Caldarelli, Teresa Disingrini, Marcella Nesi, Marco Tatò, Paola Vianello, Maria Menichincheri,